SCHEMBL23950983

SCHEMBL23950983

CC(CN)n1cnc2c(-c3cccnc3)nc(Cl)cc2c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 1/20 0.37
ADORA2A P29274 3/20 0.36
ADORA1 P30542 3/20 0.36
TBXAS1 P24557 1/20 0.36
CYP2A6 P11509 4/20 0.36
CYP2E1 P05181 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2B6 P20813 3/20 0.36
CYP2C19 P33261 3/20 0.36
CYP3A4 P08684 2/20 0.36
GRM2 Q14416 2/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
CDK5 Q00535 1/20 0.35
DYRK1A Q13627 1/20 0.35
CDK5R1 Q15078 1/20 0.35
ATR Q13535 1/20 0.34
DHPS P49366 1/20 0.34
EGLN1 Q9GZT9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23390216 0.90 KDM5B (0.37) KDM5BADORA2AADORA1TBXAS1CYP2A6
SCHEMBL23390213 0.90 KDM5B (0.37) KDM5BADORA2AADORA1TBXAS1CYP2A6
SCHEMBL23950758 0.88 PSD (0.38) KDM5BADORA2AADORA1CYP2A6CYP2E1
SCHEMBL23925644 0.85 EGLN1 (0.41) ADORA2AADORA1DYRK1ADHPSEGLN1
SCHEMBL26276200 0.83 KDM5B (0.37) KDM5BADORA2AADORA1TBXAS1CYP2A6
SCHEMBL26276204 0.83 KDM5B (0.37) KDM5BADORA2AADORA1TBXAS1CYP2A6
SCHEMBL23950999 0.82 PIM1 (0.37) KDM5BADORA2AADORA1EGLN1PIM1
SCHEMBL26276186 0.81 CYP2A6 (0.43) KDM5BADORA2AADORA1TBXAS1CYP2A6
SCHEMBL25406060 0.80 DHPS (0.40) KDM5BADORA2AADORA1TBXAS1CYP2A6
SCHEMBL25405647 0.80 DHPS (0.40) KDM5BADORA2AADORA1TBXAS1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021210970-A1 PYRIDOPYRIMIDINONE DERIVATIVES AND THEIR USE AS ARYL HYDROCARBON RECEPTOR MODULATORS DONG-A ST CO., LTD. (KR) 2021-10-21 WO disclosed