SCHEMBL23957013

SCHEMBL23957013

Cc1cnn(C)c1-c1ccc(NC[C@@H]2CC3CN(C(=O)OC(C)(C)C)C[C@H]3C2)nn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.43
BCDIN3D Q7Z5W3 1/20 0.37
NAMPT P43490 1/20 0.36
BRD4 O60885 2/20 0.36
JAK1 P23458 2/20 0.35
CDK9 P50750 2/20 0.34
CCNT1 O60563 1/20 0.34
IDO1 P14902 2/20 0.33
SPR P35270 1/20 0.33
IRAK1 P51617 1/20 0.33
JAK2 O60674 1/20 0.33
TDO2 P48775 1/20 0.33
FLT3 P36888 1/20 0.33
TYRO3 Q06418 1/20 0.33
MERTK Q12866 1/20 0.33
GAS6 Q14393 1/20 0.33
PRMT5 O14744 1/20 0.33
KDM4E B2RXH2 1/20 0.32
PKM P14618 1/20 0.32
BUB1 O43683 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29773457 1.00 NR1H2 (0.43) NR1H2BCDIN3DNAMPTBRD4JAK1
SCHEMBL23523399 1.00 NR1H2 (0.43) NR1H2BCDIN3DNAMPTBRD4JAK1
SCHEMBL23523458 0.91 NR1H2 (0.41) NR1H2BCDIN3DNAMPTJAK1SPR
SCHEMBL22797242 0.88 BCDIN3D (0.49) BCDIN3DBRD4JAK1CDK9CCNT1
SCHEMBL23932281 0.87 ACHE (0.33)
SCHEMBL20920053 0.87 ACHE (0.33)
SCHEMBL23932279 0.87 ACHE (0.33)
SCHEMBL23932284 0.87 ACHE (0.33)
SCHEMBL23523211 0.86 NR1H2 (0.38) NR1H2JAK1JAK2FLT3GPR119
SCHEMBL20936959 0.86 NR1H2 (0.38) NR1H2JAK1JAK2FLT3GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021216949-A1 CONDENSED SUBSTITUTED HYDROPYRROLES AS ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2021-10-28 WO disclosed
WO-2021216951-A1 CONDENSED SUBSTITUTED HYDROPYRROLES AS ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY (US) 2021-10-28 WO disclosed