SCHEMBL23958787

SCHEMBL23958787

CC(C)(O)c1c(F)c(-c2ccc(F)cc2)nc(C(O)(CN)C2CC2)c1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC34A1 Q06495 2/20 0.33
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32
NR3C1 P04150 1/20 0.32
HRH2 P25021 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
CFTR P13569 1/20 0.31
MAPK14 Q16539 2/20 0.31
ALOX5 P09917 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
HPGDS O60760 1/20 0.31
BRAF P15056 1/20 0.30
CDK8 P49336 1/20 0.30
CDK5 Q00535 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25686999 1.00 SLC34A1 (0.33) SLC34A1TNKSPARP1TNKS2NR3C1
SCHEMBL30007885 1.00 SLC34A1 (0.33) SLC34A1TNKSPARP1TNKS2NR3C1
SCHEMBL25687000 1.00 SLC34A1 (0.33) SLC34A1TNKSPARP1TNKS2NR3C1
SCHEMBL25686861 0.91 SLC34A1 (0.35) SLC34A1NR3C1HRH2HRH3CFTR
SCHEMBL30006977 0.91 SLC34A1 (0.35) SLC34A1NR3C1HRH2HRH3CFTR
SCHEMBL25231387 0.83 CKS1B (0.36) SLC34A1CFTRHPGDSPDK2
SCHEMBL25691242 0.83 MAPT (0.32) SLC34A1NR3C1HRH2HRH3CFTR
SCHEMBL25686730 0.82 CFTR (0.35) TNKSPARP1TNKS2CFTRALOX5
SCHEMBL28909207 0.81 CKS1B (0.32) TNKSPARP1TNKS2NR3C1HPGDS
SCHEMBL23958663 0.80 GRM2 (0.37) CFTRPDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed