SCHEMBL23958866

SCHEMBL23958866

COc1cc(C(=O)NCCO)cc2cc(C)cnc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.51
MEN1 O00255 2/20 0.51
RXFP1 Q9HBX9 1/20 0.51
SMPD1 P17405 1/20 0.46
NPC1 O15118 2/20 0.46
POLB P06746 1/20 0.45
PDE6D O43924 1/20 0.45
PDE6A P16499 1/20 0.45
PDE6G P18545 1/20 0.45
PDE6B P35913 1/20 0.45
PDE6C P51160 1/20 0.45
PDE6H Q13956 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
IRAK4 Q9NWZ3 2/20 0.43
HPGDS O60760 1/20 0.43
MMP13 P45452 1/20 0.41
BRD4 O60885 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958784 0.85 PDE4A (0.39) KMT2AMEN1RXFP1SMPD1NPC1
SCHEMBL23958791 0.84 KMT2A (0.52) KMT2AMEN1RXFP1SMPD1NPC1
SCHEMBL23905404 0.80 ATM (0.47) KMT2AMEN1NPC1POLBL3MBTL1
SCHEMBL23195851 0.79 CNR2 (0.49) POLBL3MBTL1HPGDS
SCHEMBL30007092 0.78 PARP1 (0.48) NPC1KDM4EALDH1A1HPGDSRAB9A
SCHEMBL23905400 0.77 HSD17B2 (0.49) KMT2AMEN1NPC1HPGDSRAB9A
SCHEMBL9902404 0.74 KMT2A (0.63) KMT2AMEN1RXFP1SMPD1NPC1
SCHEMBL23196217 0.72 ATM (0.44) KMT2AMEN1L3MBTL1KDM4EALDH1A1
SCHEMBL23904743 0.72 CCR1 (0.52) RXFP1KDM4EALDH1A1HPGDSMAPT
SCHEMBL30692522 0.72 CCR1 (0.42) NPC1POLBKDM4ERAB9AFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed