SCHEMBL23958892

SCHEMBL23958892

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)c(F)c(-c3ccc(F)c(F)c3)n2)C2CC2)cc2cc(C)nnc12

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSA P10619 5/20 0.35
GABRA5 P31644 3/20 0.35
CYP2C9 P11712 1/20 0.33
MAPK14 Q16539 1/20 0.33
ROCK2 O75116 3/20 0.32
ROCK1 Q13464 3/20 0.32
ABCB1 P08183 3/20 0.31
ABCC1 P33527 2/20 0.31
CNR1 P21554 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
GSK3B P49841 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25687368 1.00 CTSA (0.35) CTSAGABRA5CYP2C9MAPK14ROCK2
SCHEMBL30007118 1.00 CTSA (0.35) CTSAGABRA5CYP2C9MAPK14ROCK2
SCHEMBL25687416 0.93 CNR1 (0.37) CTSAGABRA5CYP2C9MAPK14ROCK2
SCHEMBL28909201 0.93 CNR1 (0.37) CTSAGABRA5CYP2C9MAPK14ROCK2
SCHEMBL30007246 0.93 CNR1 (0.37) CTSAGABRA5CYP2C9MAPK14ROCK2
SCHEMBL23958706 0.93 CFTR (0.36) CTSACYP2C9MAPK14ROCK2ROCK1
SCHEMBL25687411 0.93 CFTR (0.36) CTSACYP2C9MAPK14ROCK2ROCK1
SCHEMBL23958644 0.93 CFTR (0.36) CTSACYP2C9MAPK14ROCK2ROCK1
SCHEMBL30007924 0.93 CFTR (0.36) CTSACYP2C9MAPK14ROCK2ROCK1
SCHEMBL25232907 0.91 CTSA (0.34) CTSAGABRA5CYP2C9MAPK14ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed