SCHEMBL30007246

SCHEMBL30007246

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)c(F)c(-c3ccc(Cl)cc3)n2)C2CC2)cc2cc(C)nnc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.37
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.34
TP53 P04637 1/20 0.33
RHOC P08134 1/20 0.32
RHOA P61586 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CTSA P10619 2/20 0.32
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
CFTR P13569 3/20 0.31
ROCK2 O75116 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28909201 1.00 CNR1 (0.37) CNR1MAPTTHRBTP53RHOC
SCHEMBL25687416 1.00 CNR1 (0.37) CNR1MAPTTHRBTP53RHOC
SCHEMBL25687411 0.94 CFTR (0.36) CNR1MAPTCTSACFTRROCK2
SCHEMBL30007924 0.94 CFTR (0.36) CNR1MAPTCTSACFTRROCK2
SCHEMBL23958644 0.94 CFTR (0.36) CNR1MAPTCTSACFTRROCK2
SCHEMBL23958706 0.94 CFTR (0.36) CNR1MAPTCTSACFTRROCK2
SCHEMBL23958892 0.93 CTSA (0.35) CNR1MAPTCTSAROCK2ROCK1
SCHEMBL25687368 0.93 CTSA (0.35) CNR1MAPTCTSAROCK2ROCK1
SCHEMBL30007118 0.93 CTSA (0.35) CNR1MAPTCTSAROCK2ROCK1
SCHEMBL23958772 0.92 MAPT (0.35) MAPTTP53CTSAPSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed