SCHEMBL23965618

SCHEMBL23965618

CCC/C=C(\C(N)=O)c1cccc(C)c1CO

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.33
CD38 P28907 2/20 0.33
KCNH2 Q12809 1/20 0.33
KDM4E B2RXH2 2/20 0.33
GAA P10253 1/20 0.33
MYC P01106 1/20 0.33
CXCR5 P32302 5/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
HSD17B10 Q99714 1/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
PLAU P00749 2/20 0.31
F2 P00734 1/20 0.31
F10 P00742 1/20 0.31
PLG P00747 1/20 0.31
PLAT P00750 1/20 0.31
KLK1 P06870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23965593 0.87 KDM4E (0.33) CYP3A4KDM4EGAAMYCCXCR5
SCHEMBL23977989 0.84 KDM4E (0.34) CYP3A4KDM4EGAACXCR5ALDH1A1
SCHEMBL23965579 0.84 CYP3A4 (0.36) CYP3A4CD38KCNH2KDM4EGAA
SCHEMBL23965678 0.82
SCHEMBL23978149 0.76 CXCR5 (0.37) KDM4EGAACXCR5ALDH1A1HPGD
SCHEMBL30585075 0.75 CD38 (0.46) CYP3A4CD38KCNH2KDM4EGAA
SCHEMBL5963706 0.70 ALDH1A1 (0.57) CYP3A4KDM4EMYCALDH1A1HPGD
SCHEMBL6209765 0.69 CYP3A4 (0.43) CYP3A4GAAALDH1A1HSD17B10LMNA
SCHEMBL27409195 0.69 ALDH1A1 (0.55) CYP3A4KDM4EMYCALDH1A1HPGD
SCHEMBL23969498 0.68 CYP3A4 (0.38) CYP3A4KDM4EGAACXCR5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3903583-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS III BASF SE (DE) 2021-11-03 EP disclosed
EP-3903584-A1 USE OF STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI CONTAINING AN AMINO ACID SUBSTITUTION F129L IN THE MITOCHONDRIAL CYTOCHROME B PROTEIN CONFERRING RESISTANCE TO QO INHIBITORS IV BASF SE (DE) 2021-11-03 EP disclosed