SCHEMBL23966817

SCHEMBL23966817

CC(C)COc1cc2nc(Cc3n[nH]c(=O)c4ccccc34)n(COCCS(C)(C)C)c2cc1C#N

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
XDH P47989 5/20 0.37
PARP1 P09874 3/20 0.34
TNKS O95271 1/20 0.34
PARP6 Q2NL67 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
PARP3 Q9Y6F1 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
PRMT5 O14744 4/20 0.33
WDR77 Q9BQA1 4/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23915385 0.94 PARP1 (0.35) PARP1TNKSPARP6TNKS2PARP2
SCHEMBL23915393 0.85 PARP1 (0.35) PARP1TNKSPARP6TNKS2PARP2
SCHEMBL23908886 0.84 PARP1 (0.36) PARP1TNKSPARP6TNKS2PARP2
SCHEMBL23966811 0.82 PARP1 (0.36) PARP1TNKSPARP6TNKS2PARP2
SCHEMBL23915383 0.81 PARP1 (0.35) PARP1TNKSPARP6TNKS2PARP2
SCHEMBL23915442 0.76 S1PR2 (0.35)
SCHEMBL23914724 0.75 S1PR2 (0.36)
SCHEMBL23915601 0.75 S1PR2 (0.36)
SCHEMBL23915621 0.75 S1PR2 (0.41) CYP3A4CYP2C9CYP2C19
SCHEMBL23915472 0.72 XDH (0.32) XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3649119-B1 NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF FIBROSIS GALAPAGOS NV (BE) 2021-11-03 EP disclosed