SCHEMBL23967993

SCHEMBL23967993

CN[SH]1(=O)CCN(c2ccc(-c3cn(-c4ccc(F)cc4)nc3[C@@H]3CC[C@H](F)C[C@H]3C(=O)NC3(C#N)CC3)cc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 17/20 0.64
CTSB P07858 4/20 0.44
CTSS P25774 4/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968058 0.93 CTSK (0.55) CTSKCTSBCTSSKCNH2
SCHEMBL17020466 0.91 CTSK (0.77) CTSKCTSBCTSSKCNH2
SCHEMBL17008391 0.91 CTSK (0.66) CTSKCTSBCTSSKCNH2
SCHEMBL17008769 0.90 CTSK (0.63) CTSKCTSBCTSSKCNH2
SCHEMBL23968009 0.89 CTSK (0.51) CTSKCTSBCTSSKCNH2
SCHEMBL17008683 0.87 CTSK (0.82) CTSKCTSBCTSSKCNH2
SCHEMBL17008681 0.87 CTSK (0.73) CTSKCTSBCTSSKCNH2
SCHEMBL23967994 0.87 CTSK (0.66) CTSKCTSBCTSSKCNH2
SCHEMBL17008771 0.86 CTSK (0.72) CTSKCTSBCTSSKCNH2
SCHEMBL17008393 0.86 CTSK (0.73) CTSKCTSBCTSSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed