SCHEMBL23968157

SCHEMBL23968157

Fc1ccc(F)c(-n2cc(-c3ccc(N4CCSCC4)cc3)cn2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MELK Q14680 3/20 0.40
AR P10275 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 2/20 0.36
LGMN Q99538 2/20 0.36
GRM4 Q14833 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK10 P53779 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ACVR1 Q04771 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34
RXRA P19793 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
KCNH2 Q12809 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968162 0.91 MELK (0.40) MELKARL3MBTL1DRD2DRD4
SCHEMBL23968179 0.85 GRM4 (0.44) MELKDRD2DRD4DRD3LGMN
SCHEMBL23968001 0.85 MELK (0.51) MELKARL3MBTL1DRD2DRD4
SCHEMBL23968021 0.83 MELK (0.37) MELKARL3MBTL1
SCHEMBL23968168 0.83 MELK (0.46) MELKARL3MBTL1DRD2DRD4
SCHEMBL23968099 0.82 GRM4 (0.46) MELKDRD2DRD4DRD3GRM4
SCHEMBL23968105 0.80 MELK (0.39) MELKARL3MBTL1DRD2DRD4
SCHEMBL23967998 0.80 MELK (0.41) MELKARL3MBTL1DRD2DRD4
SCHEMBL23968094 0.78 MELK (0.40) MELK
SCHEMBL23968093 0.77 MAP4K4 (0.54) MELKDRD2DRD4DRD3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed