SCHEMBL23968162

SCHEMBL23968162

Fc1ccc(-n2cc(-c3ccc(N4CCSCC4)cc3)cn2)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MELK Q14680 3/20 0.40
ACKR3 P25106 1/20 0.39
ALDH1A1 P00352 2/20 0.36
ALOX15 P16050 1/20 0.36
MAPK10 P53779 1/20 0.36
HSD17B10 Q99714 1/20 0.36
AR P10275 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DRD2 P14416 2/20 0.36
DRD4 P21917 2/20 0.36
DRD3 P35462 2/20 0.36
LGMN Q99538 2/20 0.36
KDM4E B2RXH2 2/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
GRM4 Q14833 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23968157 0.91 MELK (0.40) MELKALDH1A1ALOX15MAPK10HSD17B10
SCHEMBL23968021 0.85 MELK (0.37) MELKARL3MBTL1KDM4E
SCHEMBL23968179 0.85 GRM4 (0.44) MELKDRD2DRD4DRD3LGMN
SCHEMBL23968001 0.85 MELK (0.51) MELKALDH1A1ARL3MBTL1DRD2
SCHEMBL23968168 0.83 MELK (0.46) MELKALDH1A1ARL3MBTL1DRD2
SCHEMBL23968105 0.82 MELK (0.39) MELKALDH1A1ALOX15MAPK10HSD17B10
SCHEMBL23968099 0.82 GRM4 (0.46) MELKDRD2DRD4DRD3MEN1
SCHEMBL23967998 0.80 MELK (0.41) MELKALDH1A1ARL3MBTL1DRD2
SCHEMBL19902125 0.76 NPC1 (0.46) ACKR3L3MBTL1GRM4NPC1RAB9A
SCHEMBL23968008 0.76 MELK (0.41) MELKALDH1A1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-03 EP disclosed