SCHEMBL23969467

SCHEMBL23969467

C#CCN(Cc1ccc(C)cc1)c1ccc(NC(=O)OC)c(C)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.67
CYP2C8 P10632 1/20 0.67
CYP2B6 P20813 1/20 0.67
KCNQ4 P56696 4/20 0.61
KCNQ2 O43526 1/20 0.58
KCNQ5 Q9NR82 3/20 0.58
HPGD P15428 1/20 0.44
MAPT P10636 5/20 0.43
MAPK1 P28482 3/20 0.43
GFER P55789 3/20 0.43
ALDH1A1 P00352 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
LMNA P02545 3/20 0.43
HSD17B10 Q99714 2/20 0.43
ALOX15 P16050 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HTT P42858 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18600154 0.92 CYP1A2 (0.78) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL16233333 0.84 KCNQ4 (0.86) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL15996913 0.83 KCNQ4 (0.82) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL15996918 0.82 KCNQ4 (0.70) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL19700153 0.81 KCNQ2 (0.87) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL15996931 0.81 KCNQ2 (0.83) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL16233329 0.81 CYP1A2 (0.64) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL18600189 0.81 KCNQ4 (0.68) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL18575306 0.80 CYP1A2 (1.00) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2
SCHEMBL15996895 0.80 KCNQ4 (0.70) CYP1A2CYP2C8CYP2B6KCNQ4KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3138833-B1 NOVEL KCNQ POTASSIUM CHANNEL AGONIST, AND PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI INST MATERIA MEDICA CAS (CN) 2021-11-03 EP disclosed