SCHEMBL23970774

SCHEMBL23970774

COc1nccc(Cl)c1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 2/20 0.53
HSD17B10 Q99714 1/20 0.53
POLB P06746 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
DPP4 P27487 1/20 0.41
KMO O15229 4/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
GRM4 Q14833 1/20 0.38
MTNR1A P48039 1/20 0.38
TSHR P16473 1/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30989945 1.00 ALDH1A1 (0.53) ALDH1A1KDM4EHSD17B10POLBTDP1
SCHEMBL3828695 0.84 ALDH1A1 (0.41) ALDH1A1KDM4EHSD17B10POLBTDP1
SCHEMBL7042463 0.81 CA12 (0.57) ALDH1A1KDM4EHSD17B10POLBTDP1
SCHEMBL30639556 0.80 POLB (0.43) ALDH1A1KDM4EHSD17B10POLBTDP1
SCHEMBL12794738 0.80 POLB (0.43) ALDH1A1KDM4EHSD17B10POLBTDP1
SCHEMBL27032969 0.80 POLB (0.43) ALDH1A1KDM4EHSD17B10POLBTDP1
SCHEMBL23970775 0.79 ATR (0.43) ALDH1A1KDM4EHSD17B10POLBGRM4
SCHEMBL25068658 0.79 POLB (0.42) ALDH1A1KDM4EHSD17B10POLBTDP1
SCHEMBL22090396 0.79 TDP1 (0.42) ALDH1A1KDM4EHSD17B10POLBTDP1
SCHEMBL1044983 0.79 TDP1 (0.42) ALDH1A1KDM4EHSD17B10POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222353-A1 MACROCYCLIC INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed
CN-110016025-A A kind of immunomodulator 成都先导药物开发股份有限公司 2019-07-16 CN disclosed
CN-104812755-A Pyrazolopyridine derivatives as TTX-S blockers RAQUALIA PHARMA INC 2015-07-29 CN disclosed