SCHEMBL2397111

SCHEMBL2397111

Cc1cccc(C)c1OC/C(=N\OCc1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
L3MBTL1 Q9Y468 3/20 0.44
HTR1A P08908 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
SCN4A P35499 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 2/20 0.40
SCN8A Q9UQD0 1/20 0.40
PTGER1 P34995 1/20 0.40
PTGER4 P35408 1/20 0.40
PTGER3 P43115 1/20 0.40
PTGER2 P43116 1/20 0.40
PPARG P37231 3/20 0.39
PPARA Q07869 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21325442 1.00 KMT2A (0.49) KMT2AL3MBTL1HTR1AADRA1DADRA1A
SCHEMBL2397115 1.00 KMT2A (0.49) KMT2AL3MBTL1HTR1AADRA1DADRA1A
SCHEMBL2395052 0.91 NPC1 (0.46) KMT2AL3MBTL1HTR1AADRA1DADRA1A
SCHEMBL2395055 0.91 NPC1 (0.46) KMT2AL3MBTL1HTR1AADRA1DADRA1A
SCHEMBL2390933 0.91 KMT2A (0.44) KMT2AL3MBTL1HTR1AADRA1DADRA1A
SCHEMBL2390937 0.91 KMT2A (0.44) KMT2AL3MBTL1HTR1AADRA1DADRA1A
SCHEMBL2393867 0.86 RXRA (0.50) KMT2AL3MBTL1SCN4ASMN1; SMN2NPC1
SCHEMBL2393872 0.86 RXRA (0.50) KMT2AL3MBTL1SCN4ASMN1; SMN2NPC1
SCHEMBL2393854 0.84 KMT2A (0.50) KMT2AL3MBTL1HTR1AADRA1DADRA1A
SCHEMBL2393850 0.84 KMT2A (0.50) KMT2AL3MBTL1HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed