SCHEMBL239767

SCHEMBL239767

CC(=O)Nc1ccc([N+]#N)cc1.F[B-](F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.53
SMN1; SMN2 Q16637 5/20 0.52
HTT P42858 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MEN1 O00255 4/20 0.50
ALDH1A1 P00352 2/20 0.50
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
MAPT P10636 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
CA12 O43570 1/20 0.50
BRD4 O60885 1/20 0.50
NR1I2 O75469 1/20 0.50
MB P02144 1/20 0.50
CYP1A1 P04798 1/20 0.50
CA3 P07451 1/20 0.50
CYP3A4 P08684 1/20 0.50
RARG P13631 1/20 0.50
TSHR P16473 1/20 0.50
ALOX5AP P20292 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL112275 0.93 KMT2A (0.60) KMT2ASMN1; SMN2HTTL3MBTL1MEN1
SCHEMBL31601105 0.91 SMN1; SMN2 (0.49) KMT2ASMN1; SMN2HTTL3MBTL1MEN1
Hydrochloric Acid SCHEMBL11334844 0.91 KMT2A (0.58) KMT2ASMN1; SMN2HTTL3MBTL1MEN1
SCHEMBL11877152 0.86 KMT2A (0.50) KMT2ASMN1; SMN2HTTL3MBTL1MEN1
SCHEMBL28269576 0.80 ALDH1A1 (0.51) SMN1; SMN2L3MBTL1ALDH1A1TSHRRAB9A
Acetaminophen SCHEMBL31058259 0.77 KMT2A (0.83) KMT2ASMN1; SMN2HTTL3MBTL1MEN1
SCHEMBL861674 0.76 SMN1; SMN2 (0.84) KMT2ASMN1; SMN2HTTL3MBTL1MEN1
SCHEMBL11479272 0.76 MAPT (0.45) KMT2ASMN1; SMN2L3MBTL1ALDH1A1MAPT
SCHEMBL13707197 0.75 RXFP1 (0.57) KMT2ASMN1; SMN2HTTL3MBTL1MEN1
SCHEMBL8004311 0.75 TSHR (0.37) ALDH1A1CA1CA2MAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3820629-B1 PROCESS FOR FORMING A POLYMERIC ORGANIC FILM AT THE SURFACE OF A METAL SUBSTRATE USING A GEL COMMISSARIAT ENERGIE ATOMIQUE (FR) 2024-11-27 EP claimed
EP-3077127-B1 ADHESION PRIMER FOR PAINT COMMISSARIAT ENERGIE ATOMIQUE (FR) 2018-11-14 EP claimed
US-9790370-B2 Method for preparing an organic film at the surface of a solid support under non-electrochemical conditions, solid support thus obtained and preparation kit COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2017-10-17 US claimed
US-9790371-B2 Method for preparing an organic film at the surface of a solid support under non-electrochemical conditions, solid support thus obtained and preparation kit COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2017-10-17 US claimed
US-9725602-B2 Method for preparing an organic film at the surface of a solid support under non-electrochemical conditions, solid support thus obtained and preparation kit COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2017-08-08 US claimed
EP-2077918-B1 TWO-STEP METHOD FOR FORMING ORGANIC FILMS ON ELECTRICALLY CONDUCTING SURFACES FROM AQUEOUS SOLUTIONS Commissariat à l'Energie Atomique (FR) 2017-05-17 EP claimed
EP-1989345-B1 METHOD OF FORMING ORGANIC FILMS ON ELECTRICALLY CONDUCTING OR SEMICONDUCTING SURFACES FROM AQUEOUS SOLUTIONS COMMISSARIAT L ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2015-03-11 EP claimed
US-8778165-B2 Method of forming an organic film using a gel, said gel and use thereof COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2014-07-15 US claimed
US-8709542-B2 Method for preparing an organic film at the surface of solid support under non-electrochemical conditions, solid support thus obtained and preparation kit COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2014-04-29 US claimed
EP-2155827-B1 METHOD OF FORMING AN ORGANIC FILM USING A GEL, SAID GEL AND USE THEREOF COMMISSARIAT ENERGIE ATOMIQUE (FR) 2013-07-03 EP claimed
US-20110281441-A1 Process of Localized Electrografting onto Photosensitive Semiconductor Substrates COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2011-11-17 US claimed
US-20110200790-A1 Method for Localised Electro-Grafting on Conducting or Semiconducting Substrates in the Presence of a Microelectrode COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2011-08-18 US claimed
EP-2195121-B1 METHOD OF LOCALIZED ELECTROGRAFTING ONTO PHOTOSENSITIVE SEMICONDUCTOR SUBSTRATES COMMISSARIAT ENERGIE ATOMIQUE (FR) 2011-02-23 EP claimed
US-20100310800-A1 PROCESS FOR PREPARING A METALLIZED SUBSTRATE, SAID SUBSTRATE AND USES THEREOF COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2010-12-09 US claimed
US-20100270166-A1 Method of Forming an organic Film Using a Gel, Said Gel and Use Thereof CXOMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2010-10-28 US claimed
US-20090117391-A1 METHOD FOR PREPARING AN ORGANIC FILM AT THE SURFACE OF A SOLID SUPPORT UNDER NON-ELECTROCHEMICAL CONDITIONS, SOLID SUPPORT THUS OBTAINED AND PREPARATION KIT COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2009-05-07 US claimed
US-20080193668-A1 METHOD FOR PREPARING AN ORGANIC FILM AT THE SURFACE OF A SOLID SUPPORT UNDER NON-ELECTROCHEMICAL CONDITIONS, SOLID SUPPORT THUS OBTAINED AND PREPARATION KIT COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-08-14 US claimed
US-20080152949-A1 METHOD FOR PREPARING AN ORGANIC FILM AT THE SURFACE OF A SOLID SUPPORT UNDER NON-ELECTROCHEMICAL CONDITIONS, SOLID SUPPORT THUS OBTAINED AND PREPARATION KIT COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-06-26 US claimed
US-20080145706-A1 METHOD FOR PREPARING AN ORGANIC FILM AT THE SURFACE OF SOLID SUPPORT UNDER NON-ELECTROCHEMICAL CONDITIONS, SOLID SUPPORT THUS OBTAINED AND PREPARATION KIT COMMISSARIAT A L'ENERGIE ATOMIQUE (FR) 2008-06-19 US claimed
US-20070289872-A1 Process for forming organic films on electrically conductive or semi-conductive surfaces using aqueous solutions COMMISSARIAT A L'ENERGIE ATOMIQUE 2007-12-20 US claimed