SCHEMBL23978668

SCHEMBL23978668

CN(Cc1ccccc1)C(=O)NC[C@H](CCC(=O)c1c(Cl)cc(C(=O)NCc2cccc(O)c2)cc1Cl)C(=O)OCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 1/20 0.39
ROCK2 O75116 3/20 0.36
TMEM97 Q5BJF2 3/20 0.36
SIGMAR1 Q99720 3/20 0.36
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PPARG P37231 3/20 0.35
ROCK1 Q13464 1/20 0.35
ALDH1A1 P00352 3/20 0.34
HSP90AA1 P07900 1/20 0.34
TP53 P04637 1/20 0.34
LMNA P02545 1/20 0.34
CXCR3 P49682 1/20 0.34
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26498790 0.85 MAPT (0.40) MT-CO2ROCK2TMEM97SIGMAR1NPC1
SCHEMBL23978615 0.85 MAPT (0.40) MT-CO2ROCK2TMEM97SIGMAR1NPC1
SCHEMBL23978649 0.80 ITGAL (0.44) MT-CO2ROCK2TMEM97SIGMAR1NPC1
SCHEMBL30279400 0.80 ITGAL (0.44) MT-CO2ROCK2TMEM97SIGMAR1NPC1
SCHEMBL23978549 0.80 ITGAL (0.44) MT-CO2ROCK2TMEM97SIGMAR1NPC1
SCHEMBL23978670 0.79 TMEM97 (0.45) MT-CO2ROCK2TMEM97SIGMAR1NPC1
SCHEMBL26502639 0.78 TACR1 (0.42) ROCK2TMEM97SIGMAR1NPC1RAB9A
SCHEMBL23978995 0.78 TACR1 (0.42) ROCK2TMEM97SIGMAR1NPC1RAB9A
SCHEMBL21705675 0.73 ROCK2 (0.49) MT-CO2ROCK2NPC1RAB9ASMN1; SMN2
SCHEMBL23978942 0.72 ITGB1 (0.46) TMEM97SIGMAR1NPC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed