SCHEMBL23978674

SCHEMBL23978674

CC(=O)c1c(Cl)ccc(NC(=O)Cc2cccc(Cl)c2)c1Cl

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 6/20 0.56
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
ALDH1A1 P00352 2/20 0.51
CSNK1D P48730 3/20 0.51
CACNA1G O43497 1/20 0.47
CACNA1H O95180 1/20 0.47
CACNA1C Q13936 1/20 0.47
CACNA1I Q9P0X4 1/20 0.47
MAPK8 P45983 1/20 0.46
EPHX2 P34913 1/20 0.45
POLB P06746 1/20 0.43
ANO1 Q5XXA6 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.42
TRPV1 Q8NER1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978834 0.89 KCNQ2 (0.54) KCNQ2MEN1KMT2AALDH1A1CSNK1D
SCHEMBL30336898 0.89 KCNQ2 (0.54) KCNQ2MEN1KMT2AALDH1A1CSNK1D
SCHEMBL23978894 0.88 KCNQ2 (0.54) KCNQ2MEN1KMT2AALDH1A1CSNK1D
SCHEMBL24803414 0.82 KCNQ2 (0.47) KCNQ2MEN1KMT2AALDH1A1CSNK1D
SCHEMBL26107107 0.78 KCNQ2 (0.44) KCNQ2MEN1KMT2AALDH1A1CACNA1G
SCHEMBL23978813 0.78 KCNQ2 (0.44) KCNQ2MEN1KMT2AALDH1A1CACNA1G
SCHEMBL30279468 0.78 KCNQ2 (0.44) KCNQ2MEN1KMT2AALDH1A1CACNA1G
SCHEMBL6581781 0.76 KCNQ2 (0.60) KCNQ2MEN1KMT2AALDH1A1CSNK1D
SCHEMBL23978639 0.75 KCNQ2 (0.42) KCNQ2MEN1KMT2AALDH1A1CSNK1D
SCHEMBL8279071 0.75 HPGD (0.57) KCNQ2MEN1KMT2AALDH1A1MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed