SCHEMBL23978775

SCHEMBL23978775

O=C(NC[C@H](NC(=O)c1c(Cl)cc2c(c1Cl)CCNC2)C(=O)OCc1ccccc1)NC1CCc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 4/20 0.42
ITGB2 P05107 6/20 0.38
ICAM1 P05362 6/20 0.38
ITGAL P20701 6/20 0.38
TAS1R3 Q7RTX0 2/20 0.37
TAS1R1 Q7RTX1 2/20 0.37
TAS1R2 Q8TE23 1/20 0.37
LIPG Q9Y5X9 1/20 0.36
USP2 O75604 1/20 0.35
BACE1 P56817 1/20 0.35
TAOK1 Q7L7X3 2/20 0.35
TAOK3 Q9H2K8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30083857 1.00 EPHX2 (0.42) EPHX2ITGB2ICAM1ITGALTAS1R3
SCHEMBL24803392 1.00 EPHX2 (0.42) EPHX2ITGB2ICAM1ITGALTAS1R3
SCHEMBL30279451 0.90 ITGB2 (0.46) EPHX2ITGB2ICAM1ITGALTAS1R3
SCHEMBL30083821 0.90 ITGB2 (0.46) EPHX2ITGB2ICAM1ITGALTAS1R3
SCHEMBL29019146 0.90 ITGB2 (0.46) EPHX2ITGB2ICAM1ITGALTAS1R3
SCHEMBL23978711 0.90 ITGB2 (0.46) EPHX2ITGB2ICAM1ITGALTAS1R3
SCHEMBL23978931 0.90 ITGB2 (0.46) EPHX2ITGB2ICAM1ITGALTAS1R3
SCHEMBL24803416 0.89 EPHX2 (0.40) EPHX2ITGB2ICAM1ITGALTAS1R3
SCHEMBL26502502 0.86 ITGB2 (0.44) EPHX2ITGB2ICAM1ITGAL
SCHEMBL26106382 0.86 ITGB2 (0.51) ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed