SCHEMBL29019146

SCHEMBL29019146

O=C(NCC(NC(=O)c1c(Cl)cc2c(c1Cl)CCNC2)C(=O)O)N[C@@H]1CCc2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 16/20 0.46
ICAM1 P05362 16/20 0.46
ITGAL P20701 16/20 0.46
EPHX2 P34913 2/20 0.42
ALDH1A1 P00352 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30083821 1.00 ITGB2 (0.46) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL30279451 1.00 ITGB2 (0.46) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL23978931 1.00 ITGB2 (0.46) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL23978711 1.00 ITGB2 (0.46) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL23978775 0.90 EPHX2 (0.42) ITGB2ICAM1ITGALEPHX2TAS1R3
SCHEMBL24803392 0.90 EPHX2 (0.42) ITGB2ICAM1ITGALEPHX2TAS1R3
SCHEMBL30083857 0.90 EPHX2 (0.42) ITGB2ICAM1ITGALEPHX2TAS1R3
SCHEMBL26476186 0.88 ITGB2 (0.48) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL26476093 0.88 ITGB2 (0.48) ITGB2ICAM1ITGALEPHX2ALDH1A1
SCHEMBL24803394 0.87 EPHX2 (0.48) EPHX2ALDH1A1TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916176-A Inhibitors of alpha 2 beta 1 integrin and methods of use thereof 加利福尼亚大学董事会 2023-04-04 CN disclosed