SCHEMBL23978900

SCHEMBL23978900

NC(=O)NC[C@H](NC(=O)c1c(Cl)cc(C(=O)NCc2cccc(F)c2)cc1Cl)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.45
ITGAL P20701 3/20 0.43
ITGB2 P05107 2/20 0.43
ICAM1 P05362 2/20 0.43
ITGB1 P05556 5/20 0.43
ITGA5 P08648 4/20 0.43
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
EPHX2 P34913 2/20 0.42
ALOX5 P09917 1/20 0.42
ANPEP P15144 1/20 0.41
SRC P12931 1/20 0.40
ITGA4 P13612 3/20 0.40
ROCK2 O75116 1/20 0.40
EIF4E P06730 1/20 0.40
BACE1 P56817 1/20 0.40
ITGAV P06756 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23979030 0.90 NPC1 (0.46) FOLH1ITGALITGB2ICAM1ITGB1
SCHEMBL23979033 0.88 MEN1 (0.57) ITGB1ITGA4
SCHEMBL23978899 0.86 ITGB1 (0.43) ITGALITGB1ITGA5ITGA4ROCK2
SCHEMBL3876678 0.86 ITGAL (0.48) FOLH1ITGALITGB2ICAM1ITGB1
SCHEMBL3869362 0.83 ITGAL (0.49) FOLH1ITGALITGB2ICAM1ITGB1
SCHEMBL3871439 0.80 ITGAL (0.51) ITGALITGB2ICAM1ITGB1ITGA5
SCHEMBL16286432 0.80 ITGAL (0.51) ITGALITGB2ICAM1ITGB1ITGA5
SCHEMBL30227636 0.80 ITGAL (0.51) ITGALITGB2ICAM1ITGB1ITGA5
SCHEMBL3866729 0.80 ITGAL (0.51) ITGALITGB2ICAM1ITGB1ITGA5
SCHEMBL23979041 0.80 EPHX2 (0.44) FOLH1ITGALITGB2ICAM1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed