SCHEMBL23979030

SCHEMBL23979030

NC(=O)NC[C@H](NC(=O)c1c(Cl)cc(C(=O)NCc2cccc(Cl)c2)cc1Cl)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
ITGB1 P05556 3/20 0.45
ITGA5 P08648 3/20 0.45
FOLH1 Q04609 1/20 0.42
MEN1 O00255 1/20 0.42
HCRTR1 O43613 1/20 0.42
KMT2A Q03164 1/20 0.42
C3AR1 Q16581 1/20 0.42
ITGAL P20701 2/20 0.41
ITGB2 P05107 1/20 0.41
ICAM1 P05362 1/20 0.41
APEX1 P27695 1/20 0.41
ITGA4 P13612 1/20 0.41
CTSV O60911 1/20 0.41
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978900 0.90 FOLH1 (0.45) ITGB1ITGA5FOLH1ITGALITGB2
SCHEMBL23978696 0.89 TACR1 (0.46) NPC1MEN1HCRTR1KMT2AAPEX1
SCHEMBL23978899 0.88 ITGB1 (0.43) ITGB1ITGA5C3AR1ITGALITGA4
SCHEMBL23979033 0.88 MEN1 (0.57) ITGB1MEN1KMT2AITGA4
SCHEMBL23979010 0.88 NPC1 (0.42) NPC1MEN1HCRTR1KMT2AAPEX1
SCHEMBL3866964 0.85 ITGAL (0.49) NPC1ITGB1ITGA5MEN1KMT2A
SCHEMBL23978942 0.84 ITGB1 (0.46) NPC1ITGB1ITGA5MEN1HCRTR1
SCHEMBL23978567 0.84 ITGB1 (0.46) NPC1ITGB1ITGA5MEN1HCRTR1
SCHEMBL30279319 0.84 ITGB1 (0.46) NPC1ITGB1ITGA5MEN1HCRTR1
SCHEMBL21376628 0.83 ITGB1 (0.49) ITGB1ITGA5FOLH1ITGALITGB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed