SCHEMBL23979102

SCHEMBL23979102

CC(=O)c1c(Cl)cc2c(c1Cl)CCN(C(=O)c1ccccc1)C2

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 18/20 0.58
ICAM1 P05362 18/20 0.58
ITGAL P20701 18/20 0.58
HDAC6 Q9UBN7 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10129657 0.82 ITGB2 (0.62) ITGB2ICAM1ITGALHDAC6
SCHEMBL27044184 0.80 ITGB2 (0.67) ITGB2ICAM1ITGAL
SCHEMBL18885628 0.79 ITGB2 (0.59) ITGB2ICAM1ITGALHDAC6
SCHEMBL21003874 0.78 HDAC6 (0.64) ITGB2ICAM1ITGALHDAC6
SCHEMBL18868005 0.76 ITGB2 (0.42) ITGB2ICAM1ITGALHDAC6
SCHEMBL13894069 0.75 ITGB2 (0.67) ITGB2ICAM1ITGALHDAC6
SCHEMBL13658127 0.74 ITGB2 (1.00) ITGB2ICAM1ITGAL
SCHEMBL18362337 0.74 HDAC6 (0.46) ITGB2ICAM1ITGALHDAC6
SCHEMBL13894281 0.74 ITGB2 (0.56) ITGB2ICAM1ITGALHDAC6
SCHEMBL20439976 0.74 POLB (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed