SCHEMBL23979710

SCHEMBL23979710

C=C(Cl)C(=C)C(=O)N1CCc2c(N3CCN(C(=O)OC(C)(C)C)CC3)nc(SC)nc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.41
CXCR2 P25025 1/20 0.36
GBA1 P04062 2/20 0.36
CKS1B P61024 2/20 0.36
SKP1 P63208 2/20 0.36
SKP2 Q13309 2/20 0.36
GPR119 Q8TDV5 4/20 0.35
STS P08842 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAP4K4 O95819 1/20 0.35
KIT P10721 1/20 0.35
F13A1 P00488 1/20 0.34
TGM2 P21980 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21722183 0.75 GBA1 (0.44) CXCR2GBA1CKS1BSKP1SKP2
SCHEMBL23979677 0.74 CXCR2 (0.39) CXCR2GBA1CKS1BSKP1SKP2
SCHEMBL19949022 0.72 CCNA2 (0.41) CXCR2GBA1CKS1BSKP1SKP2
SCHEMBL25771136 0.72 CXCR2 (0.38) CXCR2GBA1CKS1BSKP1SKP2
SCHEMBL23979654 0.72 GBA1 (0.39) CXCR2GBA1CKS1BSKP1SKP2
SCHEMBL19947629 0.72 ACHE (0.44) GBA1CKS1BSKP1SKP2KIT
SCHEMBL19964211 0.71 MTOR (0.45) GBA1CCNA2CDK2MAPTALDH1A1
SCHEMBL30177806 0.69 CCNA2 (0.39) CXCR2GBA1CKS1BSKP1SKP2
SCHEMBL21722244 0.69 CCNA2 (0.39) CXCR2GBA1CKS1BSKP1SKP2
SCHEMBL19616489 0.69 TMEM97 (0.46) MEN1KMT2ATLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021219072-A1 PREPARATION AND APPLICATION METHOD OF HETEROCYCLIC COMPOUND AS KRAS INHIBITOR 上海科州药物研发有限公司 (CN) 2021-11-04 WO disclosed