SCHEMBL23979724

SCHEMBL23979724

CC(C)c1nn(C)c2c(F)cccc12

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.40
ADORA1 P30542 1/20 0.40
SSTR4 P31391 9/20 0.38
KAT2B Q92831 2/20 0.32
MAPK8 P45983 1/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
EGFR P00533 1/20 0.32
SSTR1 P30872 1/20 0.32
SSTR2 P30874 1/20 0.32
SSTR3 P32745 1/20 0.32
SSTR5 P35346 1/20 0.32
TRPV4 Q9HBA0 1/20 0.32
PLK1 P53350 1/20 0.31
JAK2 O60674 1/20 0.31
BTK Q06187 1/20 0.31
ESR1 P03372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18212231 0.81 ESR1 (0.41) LMNASMN1; SMN2PLK1ESR1
SCHEMBL19954876 0.81 SSTR4 (0.50) ADORA3ADORA1SSTR4KAT2BMAPK8
SCHEMBL31582863 0.79 ADORA3 (0.40) ADORA3ADORA1SSTR4MAPK8LMNA
SCHEMBL14158503 0.78 ESR1 (0.31) ESR1
SCHEMBL13106236 0.77 SSTR4 (0.40) SSTR4KAT2BLMNAEGFRJAK2
SCHEMBL15687376 0.76 ADORA3 (0.38) ADORA3ADORA1SSTR4MAPK8SMN1; SMN2
SCHEMBL14158416 0.75 PTGER3 (0.31)
SCHEMBL16722620 0.75 SSTR4 (0.39) SSTR4KAT2BLMNAEGFRSSTR1
SCHEMBL9181361 0.75 SCN9A (0.42) SSTR4KAT2BEGFRSSTR1SSTR2
SCHEMBL20356344 0.75 ADORA3 (0.34) ADORA3ADORA1MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021219072-A1 PREPARATION AND APPLICATION METHOD OF HETEROCYCLIC COMPOUND AS KRAS INHIBITOR 上海科州药物研发有限公司 (CN) 2021-11-04 WO disclosed