SCHEMBL23989

SCHEMBL23989

Clc1ccc(COc2cccc(OBOc3cccc(OCc4ccc(Cl)cc4)c3)c2)cc1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 9/20 0.60
MAOA P21397 2/20 0.60
NR4A2 P43354 1/20 0.57
RXRA P19793 1/20 0.50
RXRB P28702 1/20 0.50
RXRG P48443 1/20 0.50
SMPD1 P17405 1/20 0.50
MEN1 O00255 1/20 0.50
MAPK1 P28482 1/20 0.50
HTT P42858 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
TLR4 O00206 1/20 0.50
TLR2 O60603 1/20 0.50
SPHK2 Q9NRA0 1/20 0.49
SPHK1 Q9NYA1 1/20 0.49
APP P05067 2/20 0.49
HPD P32754 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21409 0.85 MAOB (0.61) MAOBMAOANR4A2RXRARXRB
SCHEMBL22316 0.84 MAOB (0.66) MAOBMAOANR4A2SMPD1MEN1
SCHEMBL22564 0.82 MAOB (0.64) MAOBSMPD1TLR4TLR2SPHK2
SCHEMBL791305 0.81 MAOB (0.73) MAOBMAOANR4A2RXRARXRB
SCHEMBL4697290 0.79 APP (0.70) MAOBMAOANR4A2RXRARXRB
SCHEMBL31533129 0.79 APP (0.70) MAOBMAOANR4A2RXRARXRB
SCHEMBL4638746 0.78 MAOB (0.72) MAOBMAOANR4A2RXRARXRB
SCHEMBL13483792 0.78 MAOB (0.61) MAOBMAOANR4A2RXRARXRB
SCHEMBL13462917 0.77 MAOB (0.60) MAOBMAOANR4A2RXRARXRB
SCHEMBL23720 0.77 MAOB (0.60) MAOBAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed