SCHEMBL24013152

SCHEMBL24013152

Brc1nn(CCOC2CCCCO2)nc1Br

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
MET P08581 2/20 0.36
TGFBR1 P36897 2/20 0.33
P2RX3 P56373 7/20 0.33
TGFBR2 P37173 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24012909 0.83 KDM4C (0.42) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL12093775 0.79 KDM4C (0.38) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL9219137 0.79 KDM4C (0.40) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL24123654 0.77 KDM4C (0.42) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL20213510 0.77 KDM4C (0.42) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL28410468 0.77 KDM4C (0.37) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL28847382 0.76 KDM4C (0.39) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL10839336 0.76 KDM4C (0.38) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL26975094 0.76 KDM4C (0.38) KDM4CMEN1KMT2AL3MBTL1NPC1
SCHEMBL20519517 0.75 MET (0.44) KDM4CMEN1KMT2AL3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357269-A1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS ONCODESIGN PRECISION MEDICINE (FR) 2023-11-09 US disclosed
EP-4146658-A1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS Les Laboratoires Servier (FR) 2023-03-15 EP disclosed
WO-2021224320-A1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS LES LABORATOIRES SERVIER (FR) 2021-11-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230357269-A1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS LRRK2, RIN1, GRK3 KDM4C 2968/4885MEN1 1856/4885KMT2A 761/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.