SCHEMBL24018500

SCHEMBL24018500

Ic1ccc(N2CC3CC[C@H](C2)N3C2COC2)nc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 3/20 0.43
DRD4 P21917 3/20 0.33
HTR1A P08908 2/20 0.33
HTR2A P28223 2/20 0.33
SLC6A4 P31645 2/20 0.33
HTR7 P34969 2/20 0.33
DRD3 P35462 2/20 0.33
DRD2 P14416 2/20 0.31
HTR2C P28335 1/20 0.31
HDAC1 Q13547 1/20 0.30
EIF2AK4 Q9P2K8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20456800 1.00 MAP3K12 (0.43) MAP3K12DRD4HTR1AHTR2ASLC6A4
SCHEMBL20491963 0.94 MAP3K12 (0.38) MAP3K12DRD4HTR1AHTR2ASLC6A4
SCHEMBL20469096 0.91 MAP3K12 (0.39) MAP3K12EIF2AK4
SCHEMBL20468998 0.91 MAP3K12 (0.37) MAP3K12DRD4HTR1AHTR2ASLC6A4
SCHEMBL31447564 0.91 MAP3K12 (0.37) MAP3K12DRD4HTR1AHTR2ASLC6A4
SCHEMBL20456717 0.91 MAP3K12 (0.37) MAP3K12DRD4HTR1AHTR2ASLC6A4
SCHEMBL20456718 0.91 MAP3K12 (0.37) MAP3K12DRD4HTR1AHTR2ASLC6A4
SCHEMBL21012851 0.85 ALDH1A1 (0.33) MAP3K12DRD4HTR1AHTR2ASLC6A4
SCHEMBL24018502 0.83 MAP3K12 (0.43) MAP3K12DRD4HTR1AHTR2ASLC6A4
SCHEMBL20469202 0.83 MAP3K12 (0.46) MAP3K12DRD4HTR1AHTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3909949-A1 ATAZANAVIR (ATV) ANALOGUES FOR TREATING HIV INFECTIONS Gilead Sciences, Inc. (US) 2021-11-17 EP disclosed