SCHEMBL24019012

SCHEMBL24019012

CN[SH]1(=O)CCN(c2ccc(-c3sc(-c4cncc(F)c4)nc3[C@@H]3CCCC[C@H]3C(=O)NC3(C#N)CC3)cc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 20/20 0.65
CTSB P07858 13/20 0.46
CTSS P25774 10/20 0.46
KCNH2 Q12809 2/20 0.46
CTSL P07711 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16644716 0.93 CTSK (0.67) CTSKCTSBCTSSKCNH2CTSL
SCHEMBL18531320 0.92 CTSK (0.77) CTSKCTSBCTSSKCNH2
SCHEMBL16636416 0.91 CTSK (0.68) CTSKCTSBCTSSKCNH2
SCHEMBL16636469 0.90 CTSK (0.64) CTSKCTSBCTSSKCNH2CTSL
SCHEMBL24019032 0.88 CTSK (0.65) CTSKCTSBCTSSKCNH2
SCHEMBL16635957 0.88 CTSK (0.84) CTSKCTSBCTSSKCNH2
SCHEMBL16635956 0.88 CTSK (0.75) CTSKCTSBCTSSKCNH2
SCHEMBL16636466 0.87 CTSK (0.73) CTSKCTSBCTSSKCNH2CTSL
SCHEMBL16636414 0.87 CTSK (0.75) CTSKCTSBCTSSKCNH2
SCHEMBL16635977 0.85 CTSK (0.63) CTSKCTSBCTSSKCNH2CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3054947-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2021-11-17 EP disclosed