SCHEMBL2403402

SCHEMBL2403402

O=C(c1ccc(-c2ccccc2)cc1C(F)(F)F)N1CCC[C@H]1CN1CCCC1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 13/20 0.54
MET P08581 2/20 0.53
KCNH2 Q12809 4/20 0.53
ALK Q9UM73 1/20 0.47
OPRD1 P41143 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12393055 0.90 MET (0.49) HRH3METKCNH2ALKOPRD1
SCHEMBL12392796 0.90 MET (0.49) HRH3METKCNH2ALKOPRD1
SCHEMBL12393052 0.87 HRH3 (0.46) HRH3METKCNH2OPRD1
SCHEMBL12392794 0.87 HRH3 (0.46) HRH3METKCNH2OPRD1
SCHEMBL2343518 0.86 HRH3 (0.60) HRH3METKCNH2ALK
SCHEMBL2343522 0.86 HRH3 (0.60) HRH3METKCNH2ALK
Trifluoroacetic Acid SCHEMBL2352536 0.86 HRH3 (0.55) HRH3METKCNH2ALK
Trifluoroacetic Acid SCHEMBL2352539 0.86 HRH3 (0.55) HRH3METKCNH2ALK
SCHEMBL2345178 0.84 HRH3 (0.52) HRH3METKCNH2OPRD1
SCHEMBL2345183 0.84 HRH3 (0.52) HRH3METKCNH2OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4777974-B2 2011-09-21 JP claimed
JP-2007530698-A 2007-11-01 JP claimed
EP-1735278-A1 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND THERAPEUTIC USES ELI LILLY AND COMPANY (US) 2006-12-27 EP claimed
WO-2005097740-A1 HISTAMINE H3 RECEPTOR AGENTS, PREPARATION AND THERAPEUTIC USES ELI LILLY AND COMPANY (US) 2005-10-20 WO claimed