SCHEMBL24035652

SCHEMBL24035652

CC1(C)Cc2c(-c3cc(NC=O)ncc3Cl)cc(C#N)n2C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 14/20 0.42
CCNT1 O60563 7/20 0.42
CCNK O75909 1/20 0.38
CDK1 P06493 1/20 0.38
CDK4 P11802 1/20 0.38
CCNB1 P14635 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
MAPK8 P45983 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
CDK7 P50613 1/20 0.38
CCNH P51946 1/20 0.38
MNAT1 P51948 1/20 0.38
CSNK1G2 P78368 1/20 0.38
CDK3 Q00526 1/20 0.38
CDK6 Q00534 1/20 0.38
CDK5 Q00535 1/20 0.38
DYRK2 Q92630 1/20 0.38
CSNK1G1 Q9HCP0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25095057 0.88 CDK9 (0.37) CDK9CCNT1KDM4EALDH1A1
SCHEMBL25095132 0.87 CDK9 (0.39) CDK9CCNT1CCNKCDK1CDK4
SCHEMBL30489991 0.85 CDK9 (0.49) CDK9CCNT1CCNKCDK1CDK4
SCHEMBL25635405 0.83 CDK9 (0.39) CDK9CCNT1CCNKCDK1CDK4
SCHEMBL25095184 0.83 CDK9 (0.46) CDK9CCNT1CCNKCDK1CDK4
SCHEMBL29799769 0.82 CDK9 (0.36) CDK9CCNT1CCNKCDK1CDK4
SCHEMBL24035526 0.82 CDK9 (0.36) CDK9CCNT1CCNKCDK1CDK4
SCHEMBL24031553 0.82 CDK9 (0.36) CDK9CCNT1CCNKCDK1CDK4
SCHEMBL25095225 0.82 CDK9 (0.41) CDK9CCNT1CCNKCDK1CDK4
SCHEMBL20861661 0.80 CDK9 (0.62) CDK9CCNT1CCNKCDK1CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4141004-A1 POLYCYCLIC AMIDE DERIVATIVE AS CDK9 INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF Suzhou Alphama Biotechnology Co., Ltd. (CN) 2023-03-01 EP disclosed
WO-2021227904-A1 POLYCYCLIC AMIDE DERIVATIVE AS CDK9 INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 苏州阿尔脉生物科技有限公司 2021-11-18 WO disclosed