SCHEMBL24040264

SCHEMBL24040264

CC(C)c1cc(C(C)I)on1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.35
CHRNA1 P02708 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA7 P36544 1/20 0.33
MAPK14 Q16539 1/20 0.32
EPHX2 P34913 1/20 0.31
SCD O00767 1/20 0.30
SCD5 Q86SK9 1/20 0.30
IGF1R P08069 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22819130 0.86 GRM5 (0.41) GRM5ALDH1A1LMNASMN1; SMN2CHRNA1
SCHEMBL85820 0.83 GRM5 (0.44) GRM5ALDH1A1LMNASMN1; SMN2CHRNA1
SCHEMBL22662499 0.77 GRM5 (0.41) GRM5ALDH1A1LMNASMN1; SMN2CHRNA1
SCHEMBL11405351 0.77 GRM5 (0.44) GRM5ALDH1A1LMNASMN1; SMN2CHRNA1
SCHEMBL19135319 0.74
SCHEMBL20375480 0.74
SCHEMBL21345315 0.74 ALDH1A1 (0.41) GRM5ALDH1A1LMNASMN1; SMN2CHRNA1
SCHEMBL28297302 0.74 ALDH1A1 (0.41) GRM5ALDH1A1LMNASMN1; SMN2CHRNA1
SCHEMBL22911649 0.74 GRM5 (0.39) GRM5ALDH1A1LMNASMN1; SMN2CHRNA1
SCHEMBL1755703 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11179394-B2 Method for treating cancer using a combination of Chk1 and ATR inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2021-11-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11179394-B2 Method for treating cancer using a combination of Chk1 and ATR inhibitors CHEK1, CHEK2, ATR GRM5 4189/4885ALDH1A1 2865/4885LMNA 2309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.