SCHEMBL24049752

SCHEMBL24049752

CC(C)[C@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C)C(=O)OCc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.53
CTSB P07858 3/20 0.52
CTSK P43235 3/20 0.52
KLK5 Q9Y337 1/20 0.52
SYK P43405 1/20 0.50
CTSS P25774 4/20 0.47
PPARA Q07869 1/20 0.47
CA2 P00918 2/20 0.46
CA5A P35218 1/20 0.46
IL1RN P18510 1/20 0.46
ERAP2 Q6P179 1/20 0.46
ERAP1 Q9NZ08 1/20 0.46
CTSL P07711 2/20 0.46
CTRB1 P17538 2/20 0.46
APP P05067 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8141342 0.91 CTSK (0.56) CTSDCTSBCTSKKLK5SYK
SCHEMBL6279109 0.91 CTSK (0.56) CTSDCTSBCTSKKLK5SYK
SCHEMBL21684844 0.91 CTSK (0.56) CTSDCTSBCTSKKLK5SYK
SCHEMBL12873000 0.90 KLK5 (0.57) CTSBCTSKKLK5SYKCTSS
SCHEMBL6388701 0.90 KLK5 (0.57) CTSBCTSKKLK5SYKCTSS
SCHEMBL12214464 0.90 KLK5 (0.57) CTSBCTSKKLK5SYKCTSS
SCHEMBL24049692 0.89 SYK (0.53) CTSDCTSBCTSKKLK5SYK
SCHEMBL24049700 0.88 CTSK (0.52) CTSBCTSKKLK5SYKCTSS
SCHEMBL4904600 0.86 SYK (0.57) CTSBCTSKKLK5SYKCTSS
SCHEMBL14768567 0.86 SYK (0.57) CTSBCTSKKLK5SYKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11396497-B2 Proteasome inhibitors NEW MEXICO TECH UNIVERSITY RESEARCH PARK CORPORATION (US) 2022-07-26 US disclosed
US-20210363119-A1 PROTEASOME INHIBITORS NEW MEXICO TECH UNIVERSITY RESEARCH PARK CORPORATION 2021-11-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210363119-A1 PROTEASOME INHIBITORS TP53, CDKN1A, PSME1 CTSD 1086/4885CTSB 975/4885CTSK 646/4885
US-11396497-B2 Proteasome inhibitors TP53, CDKN1A, PSME1 CTSD 1086/4885CTSB 975/4885CTSK 646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.