SCHEMBL24070654

SCHEMBL24070654

C=NC(=C(C)C)N1CCN2C(=O)CCC2C1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SPR P35270 2/20 0.34
SCN9A Q15858 1/20 0.32
KDM5A P29375 1/20 0.32
KMT2A Q03164 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
VNN1 O95497 2/20 0.31
MEN1 O00255 1/20 0.31
BRD4 O60885 1/20 0.31
GFER P55789 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2B6 P20813 1/20 0.30
SETD2 Q9BYW2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21739460 0.80 SPR (0.37) SPRSCN9AKDM5AKMT2ANPC1
SCHEMBL21739328 0.80 SPR (0.37) SPRSCN9AKDM5AKMT2ANPC1
SCHEMBL18711619 0.79 SPR (0.40) SPRSCN9AKDM5AKMT2ANPC1
SCHEMBL10305073 0.75 SPR (0.38) SPRKDM5AKMT2ANPC1RAB9A
SCHEMBL23392344 0.73 AKR1C3 (0.39) SPRSCN9AKDM5AKMT2ANPC1
SCHEMBL23392434 0.73 AKR1C3 (0.39) SPRSCN9AKDM5AKMT2ANPC1
SCHEMBL23392436 0.73 AKR1C3 (0.39) SPRSCN9AKDM5AKMT2ANPC1
SCHEMBL16516001 0.72 SPR (0.38) SPRSCN9AKDM5AKMT2ANPC1
SCHEMBL21739380 0.72 KDM5A (0.39) SPRKDM5AKMT2ANPC1RAB9A
SCHEMBL16515572 0.72 POLB (0.46) SPRSCN9AKDM5AKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021239058-A1 FUSED TRICYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 劲方医药科技(上海)有限公司 2021-12-02 WO disclosed