SCHEMBL24075367

SCHEMBL24075367

COCCCCCOc1cc(Cl)cc(Br)c1C=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.43
ALDH1A1 P00352 3/20 0.37
USP2 O75604 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
PRKDC P78527 1/20 0.35
ERN1 O75460 1/20 0.35
PLAU P00749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16632430 0.78 PRKDC (0.52) KDM4EALDH1A1CYP1A2TDP1LMNA
SCHEMBL28821471 0.76 KDM4E (0.38) KDM4EALDH1A1USP2CYP1A2CYP2D6
SCHEMBL24075369 0.75 KDM4E (0.41) KDM4EALDH1A1USP2CYP1A2CYP2D6
SCHEMBL31028292 0.73 AAK1 (0.42) KDM4EALDH1A1CYP1A2CYP2D6LMNA
SCHEMBL19640196 0.72 LMNA (0.50) KDM4EALDH1A1USP2CYP1A2CYP2D6
SCHEMBL24075609 0.71 KDM4E (0.41) KDM4EALDH1A1USP2CYP1A2CYP2D6
SCHEMBL23658839 0.70 ERN1 (0.54) ALDH1A1TDP1LMNAHTTKMT2A
SCHEMBL24269759 0.69 ERN1 (0.46) KDM4EALDH1A1CYP1A2CYP2D6TDP1
SCHEMBL13215217 0.69 GAA (0.44) KDM4ECYP1A2CYP2D6TDP1LMNA
SCHEMBL19640183 0.68 PRKDC (0.70) KDM4EALDH1A1USP2CYP1A2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021239077-A1 MLL1 INHIBITORS AND ANTI-CANCER AGENTS NOVARTIS AG (CH) 2021-12-02 WO disclosed