SCHEMBL2408818

SCHEMBL2408818

O=C(O)C1CN(Cc2ccc(-c3cc4cc(C5CCCCC5)ccc4o3)cc2)C1.c1cc2cc(C3CCCCC3)ccc2o1

nearest known ligand 0.88

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.88
S1PR3 Q99500 8/20 0.63
S1PR5 Q9H228 4/20 0.54
S1PR4 O95977 3/20 0.54
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2476536 0.99 S1PR1 (0.86) S1PR1S1PR3S1PR5S1PR4KCNH2
SCHEMBL1602860 0.94 S1PR1 (1.00) S1PR1S1PR3S1PR5S1PR4KCNH2
SCHEMBL1602305 0.93 S1PR1 (0.98) S1PR1S1PR3S1PR5S1PR4KCNH2
SCHEMBL1603424 0.85 S1PR1 (0.83) S1PR1S1PR3S1PR5S1PR4
SCHEMBL1600910 0.83 S1PR1 (0.79) S1PR1S1PR3S1PR5S1PR4KCNH2
SCHEMBL16152955 0.82 S1PR1 (0.81) S1PR1S1PR3S1PR5S1PR4KCNH2
SCHEMBL2416672 0.82 S1PR1 (0.73) S1PR1S1PR3S1PR5S1PR4KCNH2
SCHEMBL1602550 0.82 S1PR1 (1.00) S1PR1S1PR3KCNH2
SCHEMBL1602756 0.81 S1PR1 (1.00) S1PR1S1PR3S1PR5S1PR4KCNH2
SCHEMBL12269296 0.81 S1PR1 (0.78) S1PR1S1PR3S1PR5S1PR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364976-B1 S1P receptor modulating compounds and use thereof EPIX PHARM INC (US) 2014-10-08 EP disclosed
EP-2364976-A1 S1P receptor modulating compounds and use thereof EPIX Pharmaceuticals, Inc. (US) 2011-09-14 EP disclosed