SCHEMBL2416672

SCHEMBL2416672

CC(C)CCc1ccc2oc(-c3ccc(CN4CC(C(=O)O)C4)cc3)cc2c1.CC(C)CCc1ccc2occc2c1

nearest known ligand 0.73

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.73
S1PR3 Q99500 7/20 0.73
KCNH2 Q12809 1/20 0.49
S1PR5 Q9H228 2/20 0.45
S1PR4 O95977 1/20 0.45
FFAR1 O14842 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1602626 0.94 S1PR1 (0.83) S1PR1S1PR3KCNH2S1PR5S1PR4
SCHEMBL1601177 0.85 S1PR1 (1.00) S1PR1S1PR3KCNH2S1PR5S1PR4
SCHEMBL2476536 0.83 S1PR1 (0.86) S1PR1S1PR3KCNH2S1PR5S1PR4
SCHEMBL2408818 0.82 S1PR1 (0.88) S1PR1S1PR3KCNH2S1PR5S1PR4
SCHEMBL1600903 0.82 S1PR1 (1.00) S1PR1S1PR3KCNH2S1PR5S1PR4
SCHEMBL1602228 0.82 S1PR1 (1.00) S1PR1S1PR3KCNH2S1PR5FFAR1
SCHEMBL2408724 0.81 S1PR1 (0.90) S1PR1S1PR3KCNH2S1PR5S1PR4
SCHEMBL2416119 0.81 S1PR1 (0.62) S1PR1S1PR3KCNH2S1PR5
SCHEMBL1602506 0.80 S1PR1 (0.80) S1PR1S1PR3KCNH2S1PR5S1PR4
SCHEMBL12269271 0.78 S1PR1 (0.78) S1PR1S1PR3KCNH2S1PR5S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364976-B1 S1P receptor modulating compounds and use thereof EPIX PHARM INC (US) 2014-10-08 EP disclosed
EP-2364976-A1 S1P receptor modulating compounds and use thereof EPIX Pharmaceuticals, Inc. (US) 2011-09-14 EP disclosed