SCHEMBL24101484

SCHEMBL24101484

COc1cc2cc(O)ccc2cc1C#N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.49
ESR2 Q92731 3/20 0.49
AR P10275 6/20 0.47
PGR P06401 1/20 0.47
IDH1 O75874 1/20 0.46
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
USP2 O75604 1/20 0.45
ABL1 P00519 1/20 0.44
ABCB1 P08183 1/20 0.44
BCR P11274 1/20 0.44
HTR2A P28223 1/20 0.43
MAOB P27338 1/20 0.43
MIF P14174 1/20 0.43
CA9 Q16790 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
MAP2K1 Q02750 1/20 0.41
IMPDH2 P12268 1/20 0.41
IMPDH1 P20839 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1174828 0.84 AR (0.57) ARPGRIDH1ALDH1A1KDM4E
SCHEMBL22149607 0.84 ALDH1A1 (0.53) ARPGRALDH1A1KDM4EUSP2
SCHEMBL19313480 0.83 AR (0.53) ARIDH1ALDH1A1KDM4EUSP2
SCHEMBL8500193 0.82 ESR1 (0.61) ESR1ESR2ABL1ABCB1BCR
SCHEMBL5695734 0.81 AR (0.47) ARPGRALDH1A1KDM4EUSP2
SCHEMBL15298755 0.81 AR (0.59) ARIDH1ALDH1A1KDM4EUSP2
SCHEMBL10822944 0.80 AR (0.57) ARPGRALDH1A1KDM4EUSP2
SCHEMBL3027438 0.80 ALDH1A1 (0.61) ARPGRALDH1A1KDM4EUSP2
Methane SCHEMBL28034573 0.80 ESR1 (0.59) ESR1ESR2ABL1ABCB1BCR
SCHEMBL5695670 0.78 KDM4E (0.55) ALDH1A1KDM4ECA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021249566-A1 BENZO SIX-MEMBERED RING DERIVATIVE AND USE THEREOF 山东百极地长制药有限公司 2021-12-16 WO disclosed