SCHEMBL24101702

SCHEMBL24101702

Cc1cnc(NC(=O)Cc2csc(N)n2)s1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNK O75909 2/20 0.61
DDB1 Q16531 2/20 0.61
CDK12 Q9NYV4 2/20 0.61
SMN1; SMN2 Q16637 5/20 0.55
HTT P42858 3/20 0.55
POLB P06746 1/20 0.52
ALOX12 P18054 1/20 0.49
MAPK10 P53779 1/20 0.49
GABRA5 P31644 1/20 0.49
GABRB2 P47870 1/20 0.49
HSD17B10 Q99714 1/20 0.49
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
GAA P10253 2/20 0.48
TP53 P04637 1/20 0.47
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5487408 0.84 CDK2 (0.58) CCNKDDB1CDK12SMN1; SMN2GABRA5
SCHEMBL24101425 0.84 CCNK (0.66) CCNKDDB1CDK12SMN1; SMN2HTT
SCHEMBL27569408 0.81 CCNE1 (0.53) CCNKDDB1CDK12SMN1; SMN2GABRA5
SCHEMBL24101405 0.80 CCNK (0.56) CCNKDDB1CDK12SMN1; SMN2HTT
SCHEMBL24101442 0.79 CCNK (0.81) CCNKDDB1CDK12SMN1; SMN2HTT
SCHEMBL24101742 0.79 CCNK (0.72) CCNKDDB1CDK12SMN1; SMN2HTT
SCHEMBL24101721 0.77 CCNK (0.73) CCNKDDB1CDK12SMN1; SMN2HTT
SCHEMBL24101439 0.76 CCNK (1.00) CCNKDDB1CDK12SMN1; SMN2HTT
SCHEMBL24101625 0.76 CCNK (0.78) CCNKDDB1CDK12SMN1; SMN2HTT
SCHEMBL7845357 0.76 GABRA5 (0.71) SMN1; SMN2POLBGABRA5GABRB2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021249517-A1 A MOLECULAR GLUE REGULATING CDK12-DDB1 INTERACTION TO TRIGGER CYCLIN K DEGRADATION NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2021-12-16 WO disclosed