SCHEMBL24112730

SCHEMBL24112730

Cc1ccc2c(c1)[C@@H](C)C(=O)N2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.54
EPHX2 P34913 1/20 0.43
POLB P06746 2/20 0.41
ROS1 P08922 1/20 0.40
CDK5 Q00535 1/20 0.40
ACVR1 Q04771 1/20 0.40
LRRK2 Q5S007 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
CSNK1G1 Q9HCP0 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9651557 1.00 PGR (0.54) PGREPHX2POLBROS1CDK5
SCHEMBL13091038 0.85 PGR (0.46) PGREPHX2POLBROS1CDK5
SCHEMBL24112743 0.85 PGR (0.46) PGREPHX2POLBROS1CDK5
SCHEMBL11461344 0.81 ROS1 (0.45) PGREPHX2ROS1CDK5ACVR1
SCHEMBL2263637 0.79 PGR (0.53) PGRCA12CA1CA2CA4
SCHEMBL24112727 0.79 PGR (0.53) PGRCA12CA1CA2CA4
SCHEMBL24112733 0.79 PGR (0.69) PGRPOLBKMT2AMEN1GAA
SCHEMBL29891547 0.79 PGR (0.53) PGRPOLBBRD4ALDH1A1
SCHEMBL3519770 0.79 PGR (0.53) PGRPOLBBRD4ALDH1A1
SCHEMBL948578 0.79 PGR (0.69) PGRPOLBKMT2AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021252644-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2021-12-16 WO disclosed