SCHEMBL2411570

SCHEMBL2411570

O=C(O)C1CN(Cc2ccc(-c3cc4cc(Cc5ccccc5)ccc4o3)c(F)c2)C1.O=Cc1ccc(-c2cc3cc(Cc4ccccc4)ccc3o2)c(F)c1

nearest known ligand 0.88

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.88
S1PR3 Q99500 12/20 0.88
KCNH2 Q12809 1/20 0.88

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1601733 0.94 S1PR1 (1.00) S1PR1S1PR3KCNH2
SCHEMBL1602703 0.88 S1PR1 (0.89) S1PR1S1PR3KCNH2
SCHEMBL1601354 0.88 S1PR1 (0.88) S1PR1S1PR3KCNH2
SCHEMBL1601562 0.88 S1PR1 (0.88) S1PR1S1PR3KCNH2
SCHEMBL1602248 0.87 S1PR1 (0.86) S1PR1S1PR3KCNH2
SCHEMBL4443009 0.86 S1PR1 (0.85) S1PR1S1PR3KCNH2
SCHEMBL1601119 0.86 S1PR1 (1.00) S1PR1S1PR3KCNH2
SCHEMBL1601448 0.86 S1PR1 (0.85) S1PR1S1PR3KCNH2
SCHEMBL1602394 0.86 S1PR1 (0.85) S1PR1S1PR3KCNH2
SCHEMBL1602925 0.86 S1PR1 (0.84) S1PR1S1PR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364976-B1 S1P receptor modulating compounds and use thereof EPIX PHARM INC (US) 2014-10-08 EP disclosed
EP-2364976-A1 S1P receptor modulating compounds and use thereof EPIX Pharmaceuticals, Inc. (US) 2011-09-14 EP disclosed