SCHEMBL24117147

SCHEMBL24117147

Cn1c(=O)n(CC(C)(C)O)c2cc(Oc3ccc(C(F)(F)F)cn3)ccc21

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 15/20 0.48
MAPK1 P28482 1/20 0.46
LMNA P02545 1/20 0.45
THRB P10828 1/20 0.44
SCN7A Q01118 2/20 0.44
KCNH2 Q12809 2/20 0.44
SCN10A Q9Y5Y9 1/20 0.43
SCN5A Q14524 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28356469 0.89 MAPK1 (0.47) SCN9AMAPK1LMNATHRBSCN10A
SCHEMBL28353221 0.81 SCN9A (0.50) SCN9AMAPK1SCN7AKCNH2SCN10A
SCHEMBL28356466 0.81 SCN9A (0.48) SCN9AMAPK1LMNATHRBSCN10A
SCHEMBL24116804 0.81 MAOB (0.51) SCN9AMAPK1LMNATHRBSCN7A
SCHEMBL18638520 0.76 SCN9A (0.52) SCN9AMAPK1SCN7AKCNH2SCN10A
SCHEMBL29463828 0.76 SCN9A (0.52) SCN9AMAPK1SCN7AKCNH2SCN10A
SCHEMBL29463817 0.73 SCN9A (0.54) SCN9AMAPK1SCN7AKCNH2SCN10A
SCHEMBL18638315 0.73 SCN9A (0.54) SCN9AMAPK1SCN7AKCNH2SCN10A
SCHEMBL29463882 0.70 SCN9A (0.48) SCN9AMAPK1THRBSCN7AKCNH2
SCHEMBL18638454 0.70 SCN9A (0.48) SCN9AMAPK1THRBSCN7AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110612290-A Novel benzimidazolone compounds and medicinal use thereof 大日本住友制药株式会社 2019-12-24 CN claimed
US-20210393604-A1 NOVEL BENZIMIDAZOLONE COMPOUND AND PHARMACEUTICAL USE THEREOF Sumitomo Pharma Co., Ltd. (JP) 2021-12-23 US disclosed
CN-110612290-A Novel benzimidazolone compounds and medicinal use thereof 大日本住友制药株式会社 2019-12-24 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210393604-A1 NOVEL BENZIMIDAZOLONE COMPOUND AND PHARMACEUTICAL USE THEREOF HCN4, CACNA1E, SCN1B SCN9A 55/4885MAPK1 205/4885LMNA 2589/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.