SCHEMBL24124992

SCHEMBL24124992

O=C1COc2ccc(C(=O)Nc3ccc(CNC4=CCCC=C4)cc3)cc2N1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
MAPT P10636 2/20 0.54
POLB P06746 1/20 0.54
TSHR P16473 1/20 0.52
PARP1 P09874 2/20 0.48
GAA P10253 1/20 0.48
CYP1A2 P05177 4/20 0.46
CYP3A4 P08684 4/20 0.46
CYP19A1 P11511 4/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2D6 P10635 1/20 0.46
KMT2A Q03164 1/20 0.46
TRPV1 Q8NER1 2/20 0.45
SMYD3 Q9H7B4 1/20 0.45
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25922244 0.84 PARP1 (0.71) ALDH1A1MAPTPOLBTSHRPARP1
SCHEMBL30270577 0.84 PARP1 (0.71) ALDH1A1MAPTPOLBTSHRPARP1
SCHEMBL24124197 0.80 ALDH1A1 (0.64) ALDH1A1MAPTPOLBTSHRPARP1
SCHEMBL8192718 0.78 ALDH1A1 (0.77) ALDH1A1MAPTPOLBTSHRGAA
SCHEMBL531752 0.76 ALDH1A1 (0.67) ALDH1A1MAPTPOLBTSHRPARP1
SCHEMBL14073692 0.75 ALDH1A1 (0.72) ALDH1A1MAPTPOLBTSHRGAA
SCHEMBL14072985 0.73 TSHR (0.85) ALDH1A1MAPTPOLBTSHRPARP1
SCHEMBL14073031 0.73 ALDH1A1 (0.69) ALDH1A1MAPTPOLBTSHRGAA
SCHEMBL531798 0.71 TSHR (0.74) ALDH1A1MAPTTSHRPARP1GAA
SCHEMBL24124997 0.71 ALDH1A1 (0.59) ALDH1A1MAPTPOLBTSHRPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021257544-A1 SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2021-12-23 WO disclosed