SCHEMBL2413490

SCHEMBL2413490

Cn1ncc2c(C#Cc3cccc(-c4cccc(C(F)(F)F)c4)c3)cncc21

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.41
BRD9 Q9H8M2 1/20 0.40
KCNH2 Q12809 1/20 0.39
GRIN1 Q05586 5/20 0.38
GRIN2B Q13224 5/20 0.38
FYN P06241 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
NR3C1 P04150 1/20 0.36
PGR P06401 1/20 0.36
HAO1 Q9UJM8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2419336 0.87 BRD9 (0.41) BRD9KCNH2GRIN1GRIN2BFYN
SCHEMBL1499387 0.82 NTRK1 (0.50) FYN
SCHEMBL1499372 0.80 LCK (0.54)
SCHEMBL2416274 0.78 HCRTR1 (0.43) GRM5HAO1
SCHEMBL3054046 0.77 PTGS1 (0.47)
SCHEMBL3054044 0.74 GAA (0.50) FYNNR3C1
SCHEMBL1499154 0.73 LCK (0.51) FYN
SCHEMBL1499144 0.73 NTRK1 (0.51) FYN
SCHEMBL1499307 0.72 FGFR1 (0.48)
SCHEMBL1499286 0.72 BRAF (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229389-B1 ALKYNYLARYL COMPOUNDS AND SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, METHODS OF PREPARING SAME AND USES OF SAME Bayer Pharma AG (DE) 2011-09-14 EP claimed