SCHEMBL24136199

SCHEMBL24136199

COc1cccc2cc(C)n(I)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
NQO2 P16083 4/20 0.41
CYP19A1 P11511 1/20 0.41
CCR2 P41597 1/20 0.39
NQO1 P15559 1/20 0.37
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CA4 P22748 1/20 0.37
CA7 P43166 1/20 0.37
CA14 Q9ULX7 1/20 0.37
POLB P06746 2/20 0.37
NPC1 O15118 2/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
G6PD P11413 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18000352 0.80 NQO2 (0.50) HTR2AHTR2CNQO2CYP19A1NQO1
SCHEMBL21335586 0.77 CCR2 (0.43) HTR2AHTR2CNQO2CYP19A1CCR2
SCHEMBL20989881 0.76 CYP1A2 (0.31)
SCHEMBL15971081 0.73 KDM4E (0.44) HTR2AHTR2CNQO2CYP19A1CCR2
SCHEMBL476672 0.73 HASPIN (0.41) HTR2AHTR2CNQO2CYP19A1CCR2
SCHEMBL30211234 0.72 NQO2 (0.43) HTR2AHTR2CNQO2CYP19A1CCR2
SCHEMBL20505062 0.72 HASPIN (0.46) HTR2AHTR2CNQO2CYP19A1CCR2
SCHEMBL15970972 0.72 KDM4E (0.42) HTR2AHTR2CNQO2CYP19A1CCR2
SCHEMBL24136160 0.71 HTR2C (0.39) HTR2CNQO2CYP19A1CCR2NQO1
SCHEMBL476682 0.70 HASPIN (0.44) HTR2AHTR2CNQO2CYP19A1CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3928836-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS Idorsia Pharmaceuticals Ltd (CH) 2021-12-29 EP disclosed