SCHEMBL24166758

SCHEMBL24166758

CC1CCOc2cc(I)ccc21

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 2/20 0.40
PRNP P04156 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
SRD5A1 P18405 1/20 0.33
ADRA2A P08913 3/20 0.32
ADRA2B P18089 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21933121 0.80 ADRA2A (0.41) MAP3K14ADRA2A
SCHEMBL13630579 0.80 ADRA2A (0.41) MAP3K14ADRA2A
SCHEMBL13616553 0.80 ADRA2A (0.41) MAP3K14ADRA2A
SCHEMBL24593571 0.79 ADRA2A (0.50) MAP3K14CA1CA2ADRA2A
SCHEMBL12828517 0.79 ADRA2A (0.50) MAP3K14CA1CA2ADRA2A
SCHEMBL27728300 0.79 MAP3K14 (0.65) MAP3K14CA2SRD5A1ADRA2A
SCHEMBL24866897 0.79 MAP3K14 (0.65) MAP3K14ADRA2AADRA2B
SCHEMBL24866905 0.79 MAP3K14 (0.65) MAP3K14ADRA2AADRA2B
SCHEMBL19889279 0.79 ADRA2A (0.50) MAP3K14CA1CA2ADRA2A
SCHEMBL12651543 0.79 ADRA2A (0.50) MAP3K14CA1CA2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3193601-B1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2022-01-05 EP disclosed