SCHEMBL24184663

SCHEMBL24184663

CCCOc1ccc(C#Cc2ccc(N=C=S)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.46
ACACB O00763 13/20 0.46
P2RY6 Q15077 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
LTA4H P09960 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA7 P36544 1/20 0.42
CHRNA4 P43681 1/20 0.42
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
MCHR1 Q99705 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24184660 0.93 CYP1A2 (0.46) CYP2C9ACACBP2RY6LTA4HCHRNB2
SCHEMBL24184661 0.86 NQO1 (0.50) ACACBP2RY6KMT2A
SCHEMBL9362384 0.86 CYP2C9 (0.51) CYP2C9P2RY6LTA4HCA12CA1
SCHEMBL16706066 0.84 ACACB (0.57) ACACBMEN1KMT2ALTA4HCHRNB2
SCHEMBL3434851 0.84 ACACB (0.57) ACACBMEN1KMT2ALTA4HCHRNB2
SCHEMBL26941807 0.82 P2RY6 (0.34) CYP2C9ACACBP2RY6MEN1KMT2A
SCHEMBL28275779 0.80 P2RY6 (0.40) ACACBP2RY6CHRNB2CHRNB4CHRNA3
SCHEMBL24184992 0.79 ACACB (0.43) ACACBMEN1KMT2ALTA4HCHRNB2
SCHEMBL91815 0.79 APP (0.55) ACACBP2RY6CA12CA1CA2
SCHEMBL24184976 0.79 ACACB (0.49) CYP2C9ACACBP2RY6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230313043-A1 OPTICAL COMPONENT MERCK PATENT GMBH (DE) 2023-10-05 US disclosed
US-20230313043-A1 OPTICAL COMPONENT MERCK PATENT GMBH (DE) 2023-10-05 US disclosed
WO-2022008474-A1 OPTICAL COMPONENT MERCK PATENT GMBH (DE) 2022-01-13 WO disclosed