SCHEMBL24187293

SCHEMBL24187293

CC(C)(C)OC(=O)N1CCN(c2cc(F)ccc2C=O)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.45
LMNA P02545 3/20 0.45
ALDH1A1 P00352 1/20 0.45
IDO1 P14902 1/20 0.44
TDO2 P48775 1/20 0.44
IDO2 Q6ZQW0 1/20 0.44
MAP4K4 O95819 1/20 0.44
SMARCA2 P51531 1/20 0.43
SMARCA4 P51532 1/20 0.43
PBRM1 Q86U86 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PDK2 Q15119 1/20 0.43
TP53 P04637 2/20 0.42
THRB P10828 1/20 0.42
S1PR2 O95136 1/20 0.42
GPR119 Q8TDV5 2/20 0.42
BACE1 P56817 1/20 0.41
POLB P06746 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31618908 1.00 MAPT (0.45) MAPTLMNAALDH1A1IDO1TDO2
SCHEMBL5913105 0.91 SMN1; SMN2 (0.48) MAPTLMNAALDH1A1IDO1TDO2
SCHEMBL31618922 0.91 SMN1; SMN2 (0.48) MAPTLMNAALDH1A1IDO1TDO2
SCHEMBL24187485 0.86 GPR119 (0.46) MAPTLMNAALDH1A1MAP4K4SMARCA2
SCHEMBL31618902 0.86 GPR119 (0.46) MAPTLMNAALDH1A1MAP4K4SMARCA2
SCHEMBL19582522 0.85 MAPT (0.51) MAPTLMNAALDH1A1MAP4K4SMARCA2
SCHEMBL29417615 0.85 MAPT (0.51) MAPTLMNAALDH1A1MAP4K4SMARCA2
SCHEMBL19260951 0.85 MEN1 (0.52) MAPTLMNAALDH1A1MAP4K4SMARCA2
SCHEMBL24187486 0.85 BACE1 (0.51) MAPTLMNAALDH1A1MAP4K4SMARCA2
SCHEMBL29417701 0.85 MEN1 (0.52) MAPTLMNAALDH1A1MAP4K4SMARCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115720578-A Tricyclic derivative, preparation method and medical application thereof 深圳信立泰药业股份有限公司 2023-02-28 CN disclosed
WO-2022007866-A1 FUSED TRICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATION THEREOF 深圳信立泰药业股份有限公司 2022-01-13 WO disclosed