SCHEMBL24197546

SCHEMBL24197546

N#Cc1cc(Br)cc(NCc2cccc(CO)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.45
MEF2D Q14814 1/20 0.45
NOS1 P29475 1/20 0.40
CYP19A1 P11511 1/20 0.38
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
VNN1 O95497 4/20 0.38
LRRK2 Q5S007 1/20 0.37
LMNA P02545 1/20 0.36
EGLN2 Q96KS0 2/20 0.36
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
PARP1 P09874 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HDAC1 Q13547 1/20 0.33
TDP2 O95551 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24197548 0.87 AGER (0.41) HDAC4MEF2DNOS1VNN1LRRK2
SCHEMBL24197563 0.81 HDAC4 (0.53) HDAC4MEF2DNOS1CYP19A1FFAR1
SCHEMBL24197418 0.79 POLB (0.42) FFAR1FFAR4HDAC8HDAC6PARP1
SCHEMBL24197345 0.76 AGER (0.54) CYP19A1FFAR1FFAR4HDAC8HDAC6
SCHEMBL30416299 0.76 MGAM (0.52)
SCHEMBL24197553 0.76 MGAM (0.52)
SCHEMBL24197352 0.75 CYP19A1 (0.43) CYP19A1FFAR1FFAR4VNN1HDAC8
SCHEMBL8055849 0.73 MEN1 (0.37) LMNA
SCHEMBL24197552 0.73 HDAC4 (0.40) HDAC4MEF2DNOS1CYP19A1LRRK2
SCHEMBL9454973 0.71 HDAC8 (0.57) HDAC4MEF2DFFAR1FFAR4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022011211-A1 DEOXYNOJIRIMYCIN DERIVATIVES AS GLUCOSIDASE INHIBITORS EMERGENT PRODUCT DEVELOPMENT GAITHERSBURG INC. (US) 2022-01-13 WO disclosed