SCHEMBL24200079

SCHEMBL24200079

Cc1cc(Br)c2c(c1)CCO2

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.35
CYP2A6 P11509 1/20 0.33
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
MEN1 O00255 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
RIPK1 Q13546 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL153211 0.79 AHR (0.45) PARP1CYP2A6NR3C1PGRNR3C2
SCHEMBL8011587 0.79 PARP1 (0.37) PARP1CYP2A6NR3C1PGRNR3C2
SCHEMBL13021641 0.76 PARP1 (0.40) PARP1CYP2A6PTGS1PTGS2
SCHEMBL2464027 0.76 PARP1 (0.39) PARP1CYP2A6NR3C1PGRNR3C2
SCHEMBL16004982 0.76 PARP1 (0.54) PARP1NR3C1PGRNR3C2NPSR1
SCHEMBL12330400 0.76 NOTUM (0.36) PARP1CYP2A6NR3C1PGRNR3C2
SCHEMBL23714719 0.76 PARP1 (0.42) PARP1CYP2A6NR3C1PGRNR3C2
SCHEMBL24750128 0.76 AKT1 (0.40) PARP1PTGS2NPSR1RIPK1
SCHEMBL8118010 0.76 GAA (0.39) PARP1
SCHEMBL18509016 0.76 SELL (0.39) PARP1CYP2A6NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3939658-A1 SUBSTITUTED BENZOFURAN, BENZOPYRROLE, BENZOTHIOPHENE, AND STRUCTURALLY RELATED COMPLEMENT INHIBITORS Biocryst Pharmaceuticals, Inc. (US) 2022-01-19 EP disclosed