SCHEMBL2420077

SCHEMBL2420077

c1cncc(-c2nc(C3CNCCO3)nc(C3CNCCO3)n2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.40
HTR2A P28223 1/20 0.40
ALOX15 P16050 2/20 0.39
GBA1 P04062 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
NISCH Q9Y2I1 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA5 P30532 1/20 0.39
CHRNA4 P43681 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22579073 0.78
SCHEMBL28088185 0.76 POLB (0.46) DRD2HTR2ADRD3
SCHEMBL28679348 0.76 DRD2 (0.43) DRD2DRD3
SCHEMBL30404065 0.76 DRD2 (0.55) DRD2CHRNB2CHRNA4DRD3
SCHEMBL2564441 0.76 DRD2 (0.55) DRD2CHRNB2CHRNA4DRD3
SCHEMBL27845769 0.73 DYRK1B (0.47) DRD2DRD3
SCHEMBL22122797 0.73 CYP1A1 (0.43) CYP1A2
SCHEMBL2423081 0.72 CNR2 (0.44) ALOX15KDM4EALDH1A1HPGDHSD17B10
SCHEMBL29291624 0.72 DRD2 (0.46) DRD2HTR2A
SCHEMBL28049011 0.72 DRD2 (0.36) DRD2HTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364302-A2 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES University of Basel (CH) 2011-09-14 EP claimed
WO-2010052569-A2 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES UNIVERSITY OF BASEL (CH) 2010-05-14 WO claimed